VildagliptinBasic cov ntaub ntawv
Khoom npe: | Vildagliptin |
Txhais: | Vildagliptin (NVP-LAF237); (-) - (2S) -1 - [[(3-Hydroxytricyclo [3.3.1.1 [3,7]] dec-1-yl) amino] acetyl] pyrrolidine-2-carbonitrile; 2 -PyrrolidinecarbonitChemicalbookrile, 1 - (((3-hydroxytricyclo (3.3.1.13,7) dec-1-yl) amino) acetyl) -, (2S) -; Galvus; Laf237; Unii-I6B4B2U96p; Vidagliptin (seevildagliptin); |
CAS: | 274901-16-5 |
MF: | C17H25N3O2 |
MW: | 303.4 |
VildagliptinChemical Zog
Melting taw tes | 148.0-150.0℃ |
Boiling taw tes | 531.3ºC ntawm 760 mmHg |
Yog ceev | 1.27 g / cm3 |
| Flash Point | 275.1ºC |
| Tsos | Dawb crystalline hmoov |
VildagliptinCov Khoom Qhia
Cov Khoom Qhia | Kho mob ntshav qab zib hom 2 |
Cov khoom no yog qhov ua tau zoo thiab thim rov qab tshwj xeeb kev sib tw dipeptidyl peptidase 4 (DPP-4) inhibitor. Nws qhov IC50 yog 2-3 nmol / L. Piv nrog rau lwm cov peptidases zoo sib xws, qhov tseeb IC50 ntawm DPP-4 kev cuam tshuam tau mus txog 200 μ mol / L, uas tuaj yeem zam qhov kev tiv thaiv kab mob, histopathological thiab gastrointestinal toxicity ntawm dpp-8 thiab dpp-9.
Cim npe nrov: vildagliptin cas no.274901-16-5, Suav teb, chaw tsim khoom, chaw muag khoom, Hoobkas, kev cai, lag luam wholesale
