Tofacitinib citrate Cov ncauj lus yooj yim
Khoom npe: | Tofacitinib citrate |
Txhais: | CP-690,550-10; Tasocitinib citrate; 3 - ((3R, 4R) -4-methyl-3- (methyl (7H-pyrrolo [2,3-d] pyrimidin-4-yl) amino) piperidin-1-yl ) -3-oxopropanenitrile 2-hydroxypropane-1,2,3-tricarboxylate; 2-hydroxypropane-1,2,3-tricarboxylic acid, 3 - [(3R, 4R) -4-methyl-3- [methyl (7H- pyrrolo [2,3-d] pyrimidin-4-yl) amino] piperidin-1-yl] -3-oxopropanenitrile; citro |
CAS: | 540737-29-9 |
MF: | C16H20N6O.C6H8O7 |
MW: | 504.497 |
EINECS: | 638-826-4 |
Tofacitinib citrate Lub cev thiab tshuaj tawv nqaij
Melting taw tes | 201℃ |
Boiling taw tes | Tsis muaj |
Kev Mob Cia | Chav sov |
| Flash Point | Tsis muaj |
Daim Ntawv | Dawb rau beige hmoov |
Tub sab | DMSO: soluble5mg / mL (kev daws teeb meem; sov) |
Tofacitinib citrateKev pab
Kev Siv | Jak kinase inhibitor los kho rheumatoid caj dab |
Nws siv rau cov neeg mob qog mus rau mob hnyav rau kev mob caj dab (RA) cov neeg laus cov neeg mob uas tsis muaj lus teb lossis tsis txaus siab rau kev kho mob methotrexate. Cov khoom no yog Janus kinase inhibitor, noj ob zaug ib hnub. Thaum Lub Kaum Ib Hlis 6, 2012, ib lub koomhaum tshaj lij tau tshaj tawm tias tofacitinib citrate tau txais kev pom zoo rau kev mob raum mus rau mob hnyav rau cov neeg mob cov neeg laus uas tsis tau teb lossis tsis nkag siab rau kev kho mob methotrexate. Nws tuaj yeem raug siv los ua kev kho mob ib leeg lossis hauv kev sib xyaw nrog methotrexate lossis lwm yam mob uas tsis yog roj ntsha txo cov tshuaj antirheumatic (DMARD). Cov tshuaj no yuav tsum tsis txhob siv nrog cov roj ntsha DMARDs lossis cov tshuaj tiv thaiv muaj zog (xws li azathioprine thiab cyclosporine).
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